SCHEMBL29610683

SCHEMBL29610683

CN1CCN(c2ccc(Nc3ncc(F)c(Nc4ccc5oc(=O)n(C)c5c4)n3)cn2)CC1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 5/20 0.59
JAK3 P52333 4/20 0.59
JAK2 O60674 2/20 0.59
CYP3A4 P08684 1/20 0.59
CTSC P53634 2/20 0.51
EGFR P00533 1/20 0.49
CCNT1 O60563 2/20 0.48
CCNE1 P24864 2/20 0.48
CDK2 P24941 2/20 0.48
CDK9 P50750 2/20 0.48
BRD4 O60885 5/20 0.47
SYK P43405 2/20 0.46
FLT3 P36888 2/20 0.44
BTK Q06187 2/20 0.44
WEE1 P30291 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL339911 1.00 JAK1 (0.59) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL29609910 0.90 JAK1 (0.72) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL341215 0.90 JAK1 (0.72) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL29610461 0.86 CTSC (0.54) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL340057 0.86 CTSC (0.54) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL340094 0.84 JAK1 (0.83) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL29610014 0.84 JAK1 (0.83) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL17060804 0.83 JAK1 (0.69) JAK1JAK3JAK2CYP3A4CTSC
SCHEMBL29752267 0.83 JAK1 (0.71) JAK1JAK3JAK2CYP3A4EGFR
SCHEMBL341129 0.81 JAK1 (0.68) JAK1JAK3JAK2CYP3A4CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4009974-A1 COMPOUNDS AND METHOD FOR TREATING CYTOKINE RELEASE SYNDROME Rigel Pharmaceuticals, Inc. (US) 2022-06-15 EP disclosed