Dexniguldipine

Dexniguldipine

SCHEMBL29615752

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCCN2CCC(c3ccccc3)(c3ccccc3)CC2)[C@@H]1c1cccc([N+](=O)[O-])c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 9/20 1.00
ADRA2A P08913 8/20 1.00
ADRA2B P18089 8/20 1.00
ADRA2C P18825 8/20 1.00
ADRA1D P25100 8/20 1.00
ADRA1B P35368 8/20 1.00
MAPT P10636 5/20 1.00
TDP1 Q9NUW8 4/20 1.00
MEN1 O00255 4/20 1.00
KMT2A Q03164 4/20 1.00
CYP1A2 P05177 3/20 1.00
CYP3A4 P08684 3/20 1.00
CYP2C9 P11712 3/20 1.00
CYP2C19 P33261 3/20 1.00
ABCB1 P08183 2/20 1.00
ADORA3 P0DMS8 2/20 1.00
CYP2D6 P10635 2/20 1.00
TP53 P04637 1/20 1.00
CHRM2 P08172 1/20 1.00
HTR1A P08908 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Niguldipine SCHEMBL245992 1.00 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
Dexniguldipine SCHEMBL724137 1.00 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
Niguldipine SCHEMBL245993 1.00 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
Niguldipine SCHEMBL29385244 1.00 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
Niguldipine SCHEMBL29386264 1.00 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
Niguldipine SCHEMBL3869443 0.99 ADRA1A (0.98) ADRA1AADRA2AADRA2BADRA2CADRA1D
Niguldipine SCHEMBL9001404 0.99 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
Niguldipine SCHEMBL467245 0.99 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
Dexniguldipine SCHEMBL1228966 0.99 ADRA1A (1.00) ADRA1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL9386117 0.98 ADRA1A (0.95) ADRA1AADRA2AADRA2BADRA2CADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116600799-A Pharmaceutical combination for the treatment and/or prophylaxis of diabetes 银丝佛若有限公司 2023-08-15 CN claimed
WO-2025063845-A1 DISEASE MODEL ACADEMISCH ZIEKENHUIS LEIDEN (h.o.d.n. LUMC) (NL) 2025-03-27 WO disclosed
CN-115671286-B Stereocomplex for delivery of anticancer agents 田德扬 2023-12-08 CN disclosed
EP-4126234-A1 COMPOSITIONS FOR CORONAVIRUS INFECTION TREATMENT AND/OR PREVENTION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-02-08 EP disclosed
CN-115671286-A Stereocomplex for delivery of anticancer agents 田德扬 2023-02-03 CN disclosed
CN-113260653-B Stereocomplex for delivery of anticancer agents 田德扬 2022-11-04 CN disclosed
CN-115087665-A Engineered platelets for targeted delivery of therapeutic agents JPV01有限公司 2022-09-20 CN disclosed
CN-114173797-A Product infused with cannabis with enhanced cannabinoid profile user experience 埃克索运营公司 2022-03-11 CN disclosed