SCHEMBL29616014

SCHEMBL29616014

Cc1cccc(Cl)c1NC(=O)c1cnc(N)s1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.67
LCK P06239 16/20 0.66
MAPK13 O15264 1/20 0.66
EGFR P00533 1/20 0.66
FYN P06241 1/20 0.66
HCK P08631 1/20 0.66
SRC P12931 1/20 0.66
JAK3 P52333 1/20 0.66
MAPK12 P53778 1/20 0.66
MAPK11 Q15759 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1540030 1.00 MAPK14 (0.67) MAPK14LCKMAPK13EGFRFYN
SCHEMBL4234911 0.91 MAPK14 (0.57) MAPK14LCKMAPK13EGFRFYN
SCHEMBL1539959 0.91 LCK (0.58) MAPK14LCKMAPK13EGFRFYN
SCHEMBL14416598 0.87 MAPK14 (0.70) MAPK14LCKMAPK13EGFRFYN
SCHEMBL31728413 0.87 MAPK14 (0.70) MAPK14LCKMAPK13EGFRFYN
SCHEMBL1147098 0.87 MAPK14 (0.70) MAPK14LCKMAPK13EGFRFYN
SCHEMBL29698124 0.86 MAPK14 (0.69) MAPK14LCKMAPK13EGFRFYN
SCHEMBL1539936 0.86 MAPK14 (0.69) MAPK14LCKMAPK13EGFRFYN
SCHEMBL28425094 0.85 MAPK14 (0.49) MAPK14LCKMAPK13EGFRFYN
SCHEMBL11929051 0.85 LCK (0.50) MAPK14LCKMAPK13EGFRFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118994050-A Dasatinib intermediate Synthesis method of intermediate 扬州市普林斯医药科技有限公司 2024-11-22 CN claimed
CN-114634421-A Preparation method of dasatinib intermediate 济宁晟泰药业有限公司 2022-06-17 CN claimed
CN-109796448-B Preparation process of dasatinib 山东罗欣药业集团股份有限公司 2022-05-10 CN claimed
CN-118994050-B Dasatinib intermediate Synthesis method of intermediate 扬州市普林斯医药科技有限公司 2026-03-27 CN disclosed
WO-2025231563-A1 SUBSTITUTED TRICYCLIC COMPOUNDS, COMPOSITIONS COMPRISING THEM, AND THEIR USE AS PHARMACEUTICALS UNIVERSITE DE MONTREAL (CA) 2025-11-13 WO disclosed
CN-119841819-A Degradation agent for targeting BCR-ABL and application thereof 北京大学 2025-04-18 CN disclosed
CN-118994050-A Dasatinib intermediate Synthesis method of intermediate 扬州市普林斯医药科技有限公司 2024-11-22 CN disclosed
CN-118994050-A Dasatinib intermediate Synthesis method of intermediate 扬州市普林斯医药科技有限公司 2024-11-22 CN disclosed
CN-115028678-B Bifunctional molecule based on VHL ligand-induced BCR-ABL protein degradation, and preparation method and application thereof 杭州医学院 2024-09-06 CN disclosed
EP-4326269-A1 COMPOUNDS WITH IMPROVED CARDIAC SAFETY FOR THE TREATMENT OF CANCER AND NEURODEGENERATIVE DISORDERS Oregon Health & Science University (US) 2024-02-28 EP disclosed
WO-2022225972-A1 COMPOUNDS WITH IMPROVED CARDIAC SAFETY FOR THE TREATMENT OF CANCER AND NEURODEGENERATIVE DISORDERS OREGON HEALTH & SCIENCE UNIVERSITY (US) 2022-10-27 WO disclosed
CN-115028678-A Bifunctional molecule based on BCR-ABL protein degradation induced by VHL ligand and preparation method and application thereof 杭州医学院 2022-09-09 CN disclosed
CN-111212833-B Phenylpyridine derivatives and pharmaceutical compositions containing the same 株式会社大熊制药 2022-09-06 CN disclosed
CN-114634421-A Preparation method of dasatinib intermediate 济宁晟泰药业有限公司 2022-06-17 CN disclosed
CN-109796448-B Preparation process of dasatinib 山东罗欣药业集团股份有限公司 2022-05-10 CN disclosed
CN-109796448-B Preparation process of dasatinib 山东罗欣药业集团股份有限公司 2022-05-10 CN disclosed