SCHEMBL29616591

SCHEMBL29616591

N=C(NO)c1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.44
ALDH1A1 P00352 4/20 0.42
MAPT P10636 3/20 0.42
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
SORT1 Q99523 1/20 0.40
AVPR2 P30518 1/20 0.40
GPR27 Q9NS67 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
CES2 O00748 2/20 0.40
LMNA P02545 2/20 0.38
MEN1 O00255 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TRPV1 Q8NER1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23148979 1.00 PDE2A (0.44) PDE2AALDH1A1MAPTJAK2JAK1
SCHEMBL28571714 0.80 GPR27 (0.55) ALDH1A1MAPTJAK2JAK1TYK2
SCHEMBL17814063 0.79 PDE2A (0.46) PDE2AALDH1A1MAPTSORT1AVPR2
SCHEMBL29616566 0.76 SMN1; SMN2 (0.50) ALDH1A1MAPTJAK2JAK1TYK2
SCHEMBL4145427 0.76 SMN1; SMN2 (0.50) ALDH1A1MAPTJAK2JAK1TYK2
SCHEMBL4357462 0.75 AVPR2 (0.50) PDE2AALDH1A1MAPTJAK2JAK1
SCHEMBL4680773 0.74 FLT1 (0.43) ALDH1A1LMNAMEN1HTTKMT2A
SCHEMBL3276332 0.74 HSD17B10 (0.46) ALDH1A1MAPTCES2LMNAHTT
SCHEMBL4511425 0.73 P2RX1 (0.53) ALDH1A1MAPTJAK2JAK1TYK2
SCHEMBL1818435 0.73 KDM4E (0.62) PDE2AALDH1A1SORT1AVPR2GPR27

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114401968-A Novel heterocyclic monoacylglycerol lipase (MAGL) inhibitors 豪夫迈·罗氏有限公司 2022-04-26 CN disclosed