SCHEMBL29622100

SCHEMBL29622100

Cc1cc(N)cc(C)c1Oc1ccc2c(c1)C1(CCCC1)C(=O)N2

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PGR P06401 12/20 0.43
MAPK14 Q16539 5/20 0.42
PDE4A P27815 3/20 0.40
PDE4B Q07343 3/20 0.40
PDE4C Q08493 3/20 0.40
PDE4D Q08499 3/20 0.40
PDE3B Q13370 3/20 0.40
PDE3A Q14432 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29076828 0.98 PGR (0.43) PGRMAPK14PDE4APDE4BPDE4C
SCHEMBL29621962 0.98 PGR (0.43) PGRMAPK14PDE4APDE4BPDE4C
SCHEMBL29621937 0.95 PGR (0.40) PGRMAPK14PDE4APDE4BPDE4C
SCHEMBL29621927 0.95 PGR (0.40) PGRMAPK14PDE4APDE4BPDE4C
SCHEMBL29621911 0.84 PGR (0.55) PGRMAPK14PDE4APDE4BPDE4C
SCHEMBL29622023 0.83 PGR (0.48) PGRPDE4APDE4BPDE4CPDE4D
SCHEMBL29621965 0.81 PGR (0.52) PGRMAPK14PDE4APDE4BPDE4C
SCHEMBL29076750 0.81 PGR (0.52) PGRMAPK14PDE4APDE4BPDE4C
SCHEMBL28530057 0.80 PGR (0.46) PGR
SCHEMBL29622021 0.80 PGR (0.46) PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4240722-A1 OXINDOLES AND METHODS OF USE THEREOF Aligos Therapeutics, Inc. (US) 2023-09-13 EP disclosed
WO-2022099066-A1 OXINDOLES AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2022-05-12 WO disclosed