SCHEMBL29622993

SCHEMBL29622993

O=C(O)c1cccc(Oc2ccnc3ccccc23)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.56
LOXL2 Q9Y4K0 1/20 0.50
MRGPRX4 Q96LA9 1/20 0.49
KDR P35968 3/20 0.48
BRAF P15056 1/20 0.48
MAPK14 Q16539 1/20 0.48
TNNI3K Q59H18 1/20 0.48
GPBAR1 Q8TDU6 1/20 0.48
CYSLTR1 Q9Y271 1/20 0.48
NR4A2 P43354 1/20 0.47
KMO O15229 1/20 0.46
MIF P14174 2/20 0.45
AR P10275 1/20 0.45
F2 P00734 1/20 0.45
F10 P00742 1/20 0.45
TTR P02766 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22972144 1.00 AKR1C3 (0.56) AKR1C3LOXL2MRGPRX4KDRBRAF
SCHEMBL29622884 0.88 TNKS (0.51) KDRBRAFMAPK14TNNI3KF2
SCHEMBL24724269 0.88 MEN1 (0.58) KDRBRAFMAPK14TNNI3KGPBAR1
SCHEMBL24724243 0.88 TNKS (0.51) KDRBRAFMAPK14TNNI3KF2
SCHEMBL29622922 0.88 TNKS (0.51) KDRBRAFMAPK14TNNI3KF2
SCHEMBL24724242 0.85 KDR (0.50) KDRBRAFMAPK14TNNI3KAR
SCHEMBL7237590 0.83 TTR (0.54) AKR1C3KDRTTR
SCHEMBL22972360 0.83 LOX (0.62) LOXL2AR
SCHEMBL22972145 0.83 DDR2 (0.54) KDRBRAFMAPK14TNNI3K
SCHEMBL30050285 0.83 DDR2 (0.54) KDRBRAFMAPK14TNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114391009-A Quinoline derivatives as protein kinase inhibitors BCI制药公司 2022-04-22 CN disclosed