SCHEMBL29623536

SCHEMBL29623536

COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OC1CCN(C)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 1.00
KDR P35968 5/20 0.75
FLT1 P17948 2/20 0.75
FGFR1 P11362 1/20 0.75
ERBB2 P04626 4/20 0.74
EPHB4 P54760 4/20 0.74
EPHA2 P29317 3/20 0.74
AURKA O14965 1/20 0.73
INSR P06213 1/20 0.73
FBP1 P09467 1/20 0.73
PDGFRB P09619 1/20 0.73
FLT4 P35916 1/20 0.73
CLK1 P49759 1/20 0.73
TEK Q02763 1/20 0.73
AURKB Q96GD4 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL185721 1.00 EGFR (1.00) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL12743397 0.96 EGFR (0.92) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL10285954 0.91 EGFR (0.84) EGFRKDRERBB2EPHB4EPHA2
SCHEMBL4416173 0.91 EGFR (0.84) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL4096274 0.91 EGFR (0.84) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL10285957 0.91 EGFR (0.84) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL1446584 0.91 EGFR (0.84) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL1446182 0.91 EGFR (0.83) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL29623562 0.91 EGFR (0.83) EGFRKDRFLT1FGFR1ERBB2
SCHEMBL210910 0.91 EGFR (0.83) EGFRKDRFLT1FGFR1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110840847-B Pharmaceutical compositions for the treatment of cystic fibrosis transmembrane conductance regulator mediated diseases 沃泰克斯药物股份有限公司 2022-07-29 CN disclosed
CN-110713489-B Heteroaryl SYK inhibitors 勃林格殷格翰国际有限公司 2022-05-31 CN disclosed
CN-110183440-B Heteroaryl SYK inhibitors 勃林格殷格翰国际有限公司 2022-04-22 CN disclosed