SCHEMBL29624095

SCHEMBL29624095

CCCc1cc(F)c(F)c(C(=O)c2ccc3ncc(N4CCOCC4)nc3c2)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.42
CDK6 Q00534 2/20 0.42
PIK3CD O00329 5/20 0.40
PIK3CA P42336 5/20 0.40
PIK3CB P42338 5/20 0.40
PIK3CG P48736 5/20 0.40
MTOR P42345 4/20 0.40
FGFR2 P21802 1/20 0.40
FGFR3 P22607 1/20 0.40
NPC1 O15118 1/20 0.39
SHMT2 P34897 2/20 0.39
PRKDC P78527 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
DGAT1 O75907 1/20 0.38
SOAT1 P35610 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14741376 0.86 CDK6 (0.40) HPGDCDK6PIK3CDPIK3CAPIK3CB
SCHEMBL14829458 0.85 HPGD (0.46) HPGDCDK6PIK3CDPIK3CAPIK3CB
SCHEMBL14716084 0.85 HDAC3 (0.45) HPGDCDK6PIK3CDPIK3CAPIK3CB
SCHEMBL20749378 0.83 CDK6 (0.41) HPGDCDK6PIK3CDPIK3CAPIK3CB
SCHEMBL29623952 0.83 CDK6 (0.41) HPGDCDK6PIK3CDPIK3CAPIK3CB
SCHEMBL14715976 0.82 CDK6 (0.39) HPGDCDK6PIK3CDPIK3CAPIK3CB
Uplarafenib SCHEMBL14716189 0.82 BRAF (0.51) HPGDCDK6PIK3CDPIK3CAPIK3CB
SCHEMBL29623943 0.82 CDK6 (0.39) HPGDCDK6PIK3CDPIK3CAPIK3CB
Uplarafenib SCHEMBL29623930 0.82 BRAF (0.51) HPGDCDK6PIK3CDPIK3CAPIK3CB
SCHEMBL20246640 0.81 HPGD (0.44) HPGDCDK6PIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4255434-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Neupharma, Inc. (US) 2023-10-11 EP claimed
WO-2022119905-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA, INC (US) 2022-06-09 WO claimed