SCHEMBL2962478

SCHEMBL2962478

Cn1c(C2CCOCC2)nc(C(=O)NC(=O)NCc2ccccc2N2CCCCS2(=O)=O)c(O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CALCA P06881 13/20 0.39
AADAT Q8N5Z0 1/20 0.38
LIPG Q9Y5X9 2/20 0.37
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2955395 0.96 CALCA (0.38) CALCAAADATLIPGCYP3A4CYP2C19
SCHEMBL13243792 0.94 CALCA (0.44) CALCAAADATLIPGCYP2C9
SCHEMBL2967365 0.90 CALCA (0.41) CALCAAADATCYP2C9
SCHEMBL13243787 0.90 CALCA (0.43) CALCAAADATLIPGCYP2C9
SCHEMBL2957301 0.86 CALCA (0.40) CALCACYP2C9
SCHEMBL13243791 0.84 CALCA (0.46) CALCAAADATCYP2C9
SCHEMBL13243788 0.80 CALCA (0.45) CALCACYP3A4CYP2C9
SCHEMBL13917566 0.75 CALCA (0.44) CALCALIPGCYP3A4CYP2C19CYP2C9
SCHEMBL13917556 0.74 CALCA (0.46) CALCALIPGCYP3A4CYP2C19CYP2C9
SCHEMBL3840245 0.73 CALCA (0.43) CALCALIPGCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7763630-B2 pyrimidinone compounds such as N-(4-Fluorobenzyl)-5-hydroxy-1-methyl-6-oxo-2-(tetrahydrofuran-3-yl)-1,6-dihydropyrimidine-4-carboxamide, used for treating human immunodeficiency virus (HIV) and acquired immune deficiency syndrome (AIDS) BRISTOL-MYERS SQUIBB COMPANY (US) 2010-07-27 US claimed
US-20080306051-A1 HIV Integrase Inhibitors BRISTOL-MYERS SQUIBB COMPANY 2008-12-11 US claimed
US-7763630-B2 pyrimidinone compounds such as N-(4-Fluorobenzyl)-5-hydroxy-1-methyl-6-oxo-2-(tetrahydrofuran-3-yl)-1,6-dihydropyrimidine-4-carboxamide, used for treating human immunodeficiency virus (HIV) and acquired immune deficiency syndrome (AIDS) BRISTOL-MYERS SQUIBB COMPANY (US) 2010-07-27 US disclosed
US-20080306051-A1 HIV Integrase Inhibitors BRISTOL-MYERS SQUIBB COMPANY 2008-12-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306051-A1 HIV Integrase Inhibitors TYMP, IMPDH1, UNG CALCA 2954/4885AADAT 1332/4885LIPG 4508/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.