SCHEMBL29625543

SCHEMBL29625543

CC(C)n1cc(C(N)=O)c(=O)n(-c2ccccc2)c1=O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
MAPK1 P28482 1/20 0.43
MET P08581 2/20 0.41
TYRO3 Q06418 5/20 0.40
MERTK Q12866 4/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GSK3A P49840 2/20 0.38
GSK3B P49841 2/20 0.38
PGR P06401 1/20 0.37
AXL P30530 1/20 0.36
RIPK2 O43353 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31614377 0.99 KMT2A (0.47) KMT2AMAPK1METTYRO3MERTK
SCHEMBL14969331 0.88 KMT2A (0.44) KMT2AMETTYRO3MERTKKDM4E
SCHEMBL30030688 0.87 KMT2A (0.39) KMT2AMAPK1METTYRO3MERTK
SCHEMBL19398124 0.87 KDM4E (0.45) KMT2AMETTYRO3MERTKKDM4E
SCHEMBL30030585 0.86 AXL (0.41) KMT2AMAPK1METTYRO3MERTK
SCHEMBL29536487 0.86 AXL (0.47) METTYRO3MERTKAXL
Hydrochloric Acid SCHEMBL30297740 0.85 AXL (0.47) METTYRO3MERTKAXL
SCHEMBL29626219 0.84 PDE4A (0.42) KMT2AMAPK1METMERTKGSK3A
SCHEMBL29626208 0.84 AXL (0.48) KMT2AMETTYRO3MERTKAXL
SCHEMBL30672108 0.84 TYRO3 (0.43) KMT2AMETTYRO3AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114456175-B Pyrrolotriazine compounds as TAM inhibitors 因赛特公司 2024-09-03 CN claimed
EP-3436461-B1 PYRROLOTRIAZINE COMPOUNDS AS TAM INHIBITORS INCYTE CORP (US) 2023-11-01 EP claimed
CN-114456176-A Pyrrolotriazine compounds as TAM inhibitors 因赛特公司 2022-05-10 CN claimed
CN-114456175-B Pyrrolotriazine compounds as TAM inhibitors 因赛特公司 2024-09-03 CN disclosed
CN-114456176-B Pyrrolotriazine compounds as TAM inhibitors 因赛特公司 2024-08-30 CN disclosed
EP-3436461-B1 PYRROLOTRIAZINE COMPOUNDS AS TAM INHIBITORS INCYTE CORP (US) 2023-11-01 EP disclosed
CN-114456175-A Pyrrolotriazine compounds as TAM inhibitors 因赛特公司 2022-05-10 CN disclosed
CN-114456176-A Pyrrolotriazine compounds as TAM inhibitors 因赛特公司 2022-05-10 CN disclosed