SCHEMBL29627424

SCHEMBL29627424

O=c1[nH]cnc2c1ccn2-c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 2/20 0.45
KDM4B O94953 2/20 0.45
KDM5C P41229 2/20 0.45
KDM5B Q9UGL1 2/20 0.45
KDM4C Q9H3R0 1/20 0.45
KDM3A Q9Y4C1 1/20 0.45
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2A6 P11509 1/20 0.42
LDHA P00338 1/20 0.41
ALDH1A1 P00352 2/20 0.41
SRC P12931 1/20 0.41
AR P10275 1/20 0.40
MAPT P10636 2/20 0.40
PI4KA P42356 1/20 0.39
PI4K2B Q8TCG2 1/20 0.39
PI4K2A Q9BTU6 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
HTT P42858 1/20 0.39
ELANE P08246 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20971254 1.00 KDM4A (0.45) KDM4AKDM4BKDM5CKDM5BKDM4C
SCHEMBL20971053 0.85 SRC (0.55) LDHAALDH1A1SRCMAPTHTT
SCHEMBL20971301 0.84 KDM4A (0.45) KDM4AKDM4BKDM5CKDM5BKDM4C
SCHEMBL20971362 0.79 PARP1 (0.42) KDM4AKDM4BKDM5CKDM5BKDM4C
SCHEMBL32668797 0.79 HTT (0.51) KDM4AKDM4BKDM5CKDM5BKDM4C
SCHEMBL20971017 0.79 MAPT (0.51) ALDH1A1SRCMAPTPARP1HPGD
SCHEMBL20971046 0.78 LMNA (0.58) ALDH1A1SRCMAPTHTTPARP1
SCHEMBL20971117 0.78 KMT2A (0.50) SRCMAPTPI4KAPI4K2BPI4K2A
SCHEMBL17868975 0.78 PIM1 (0.46) ALDH1A1SRCMAPTPARP1PDPK1
SCHEMBL29627437 0.78 PARP1 (0.46) ALDH1A1SRCMAPTPARP1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563094-B (hetero) aryl-substituted piperidinyl derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2022-03-18 CN claimed
CN-109563094-B (hetero) aryl-substituted piperidinyl derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2022-03-18 CN disclosed