SCHEMBL29627707

SCHEMBL29627707

C#Cn1ncc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
RECQL P46063 1/20 0.43
KMO O15229 1/20 0.42
SLC22A12 Q96S37 1/20 0.37
ELANE P08246 1/20 0.37
PDE10A Q9Y233 2/20 0.37
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
DAO P14920 1/20 0.36
ASAH1 Q13510 2/20 0.35
TFPI2 P48307 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16874288 0.89 CYP1A2 (0.37) CYP1A2RECQLKMOSLC22A12ELANE
SCHEMBL953069 0.81 CYP1A2 (0.44) CYP1A2RECQLKMOSLC22A12ELANE
SCHEMBL5748095 0.79 CYP1A2 (0.51) CYP1A2RECQLKMOSLC22A12ELANE
SCHEMBL30419498 0.79 CYP1A2 (0.51) CYP1A2RECQLKMOSLC22A12ELANE
SCHEMBL28206607 0.73 CYP1A2 (0.39) CYP1A2RECQLKMOSLC22A12ELANE
SCHEMBL31690942 0.72 CYP11B1 (0.38) CYP1A2RECQLKMOSLC22A12ELANE
SCHEMBL276287 0.71 RECQL (0.47) CYP1A2RECQLKMOSLC22A12ELANE
SCHEMBL9934408 0.71 RECQL (0.61) CYP1A2RECQLKMODDB1CRBN
SCHEMBL30755148 0.71 RECQL (0.56) CYP1A2RECQLKMOPDE10AADRA2A
SCHEMBL4287336 0.71 RECQL (0.56) CYP1A2RECQLKMOPDE10AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4003340-A2 ETHYNYLHETEROCYCLES AS RHO-ASSOCIATED COILED-COIL KINASE (ROCK) INHIBITORS Angion Biomedica Corp. (US) 2022-06-01 EP claimed
EP-4003340-A2 ETHYNYLHETEROCYCLES AS RHO-ASSOCIATED COILED-COIL KINASE (ROCK) INHIBITORS Angion Biomedica Corp. (US) 2022-06-01 EP disclosed