SCHEMBL29627975

SCHEMBL29627975

CC1CN(c2ccc3c(c2)CN(c2nccc(-c4nccc(C#Cc5ccc6[nH]ncc6c5)n4)n2)C3)CCO1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 18/20 0.41
ROCK1 Q13464 8/20 0.38
TMEM97 Q5BJF2 1/20 0.34
IDH1 O75874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29627923 0.87 ROCK2 (0.45) ROCK2ROCK1TMEM97
SCHEMBL29627719 0.82 ROCK2 (0.53) ROCK2ROCK1TMEM97
SCHEMBL29640423 0.82 ROCK2 (0.56) ROCK2ROCK1TMEM97
SCHEMBL29627761 0.82 ROCK2 (0.56) ROCK2ROCK1TMEM97
SCHEMBL29627940 0.82 ROCK2 (0.48) ROCK2ROCK1TMEM97
SCHEMBL29627730 0.82 ROCK2 (0.61) ROCK2ROCK1TMEM97
SCHEMBL29627828 0.81 ROCK2 (0.58) ROCK2ROCK1
SCHEMBL29627716 0.80 ROCK2 (0.46) ROCK2ROCK1TMEM97
SCHEMBL29640512 0.80 ROCK2 (0.46) ROCK2ROCK1TMEM97
SCHEMBL29640483 0.80 ROCK2 (0.46) ROCK2ROCK1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4003340-A2 ETHYNYLHETEROCYCLES AS RHO-ASSOCIATED COILED-COIL KINASE (ROCK) INHIBITORS Angion Biomedica Corp. (US) 2022-06-01 EP disclosed
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed