SCHEMBL29628279

SCHEMBL29628279

Cc1c(C2CO2)ccc(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.36
TAAR1 Q96RJ0 2/20 0.35
CYP2D6 P10635 1/20 0.35
HDAC4 P56524 1/20 0.34
BRD4 O60885 1/20 0.33
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
TSHR P16473 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA7 P36544 1/20 0.30
CHRNA4 P43681 1/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4306696 0.81 TSHR (0.34) HTR2CHTR2BTSHRCHRNB2CHRNB4
SCHEMBL17141386 0.80 TSHR (0.40) TAAR1CYP2D6HTR2CHTR2BTSHR
SCHEMBL13027719 0.77 KCNJ1 (0.44)
SCHEMBL286934 0.77 KCNJ1 (0.44)
SCHEMBL14723162 0.77 AR (0.41) CYP11B1CYP11B2
SCHEMBL20819598 0.76 CYP2D6 (0.35) TAAR1CYP2D6HTR2CHTR2BNOS3
SCHEMBL20833596 0.75 HTR2C (0.49) TAAR1CYP2D6HTR2CHTR2BTSHR
SCHEMBL7055104 0.75 HTR2C (0.49) TAAR1CYP2D6HTR2CHTR2BTSHR
SCHEMBL17865235 0.72 BRD4 (0.38) CYP2D6BRD4HTR2CHTR2BCHRNB2
SCHEMBL10779356 0.71 HTR2C (0.49) TAAR1CYP2D6HTR2CHTR2BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3997096-A1 NEW HETEROCYCLIC COMPOUNDS F. Hoffmann-La Roche AG (CH) 2022-05-18 EP disclosed