SCHEMBL29629115

SCHEMBL29629115

O=C1c2ccccc2C(=O)N1Cc1cc(Cl)ccc1Br

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 12/20 0.52
CYP1B1 Q16678 2/20 0.50
TYR P14679 1/20 0.46
CASP3 P42574 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2558741 1.00 GRM5 (0.52) GRM5CYP1B1TYRCASP3CA12
SCHEMBL9478240 0.85 GRM5 (0.55) GRM5TYRCASP3
SCHEMBL3729290 0.84 GRM5 (0.54) GRM5TYRCASP3
SCHEMBL14338959 0.81 RPS6KA2 (0.53) GRM5CYP1B1TYRCASP3CA12
SCHEMBL6076008 0.81 GRM5 (0.62) GRM5CASP3CA12CA1CA2
SCHEMBL18669095 0.81 RPS6KA2 (0.53) GRM5CYP1B1TYRCASP3
SCHEMBL11081773 0.81 MAPT (0.58) GRM5TYRCASP3CA12CA1
SCHEMBL6095022 0.80 TYR (0.64) GRM5CYP1B1TYRCASP3CA12
SCHEMBL5957957 0.78 TP53 (0.58) GRM5CASP3
SCHEMBL8311470 0.78 ALDH1A1 (0.52) GRM5CASP3CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621135-B LPA1 small molecule antagonist 上海拓界生物医药科技有限公司 2024-01-30 CN disclosed
CN-114621135-A LPA1 small molecule antagonist 上海拓界生物医药科技有限公司 2022-06-14 CN disclosed