SCHEMBL29629416

SCHEMBL29629416

NC(=O)c1cccc(C(F)(F)F)c1-c1cc[nH]n1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.43
PDK2 Q15119 1/20 0.41
SCN9A Q15858 2/20 0.37
AURKA O14965 2/20 0.37
RPS6KB1 P23443 1/20 0.37
AURKB Q96GD4 1/20 0.37
FABP4 P15090 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
CD38 P28907 2/20 0.35
CYP3A4 P08684 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
PDPK1 O15530 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7163549 0.81 PARP1 (0.40) PARP1PDK2AURKAKEAP1NFE2L2
SCHEMBL3422877 0.80 PARP1 (0.41) PARP1AURKALMNACD38CYP3A4
SCHEMBL3421071 0.78 PARP1 (0.40) PARP1AURKALMNAKEAP1NFE2L2
SCHEMBL18398143 0.78 JAK2 (0.31) SCN9A
SCHEMBL18398127 0.78 PARP1 (0.34) PARP1
SCHEMBL29543435 0.78 PARP1 (0.41) PARP1PDK2SCN9AAURKAKEAP1
SCHEMBL15904410 0.77 CTNNB1 (0.48) PARP1PDK2SCN9AAURKARPS6KB1
SCHEMBL18398075 0.77 PARP1 (0.35) PARP1LMNAGAA
SCHEMBL8132468 0.77 PARP1 (0.47) PARP1PDK2SCN9AAURKARPS6KB1
SCHEMBL3419413 0.76 PARP1 (0.44) PARP1AURKARPS6KB1KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3994138-A1 ESTROGEN-RELATED RECEPTOR ALPHA (ERRalpha) MODULATORS Lead Pharma Holding B.V. (NL) 2022-05-11 EP claimed