SCHEMBL29633203

SCHEMBL29633203

COc1cc(Oc2ccnc3ccccc23)cc(C(=O)NCc2ccccc2OC)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 2/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
HPGD P15428 4/20 0.57
GAA P10253 2/20 0.57
MAPT P10636 2/20 0.50
POLB P06746 3/20 0.49
HTT P42858 2/20 0.49
DDR2 Q16832 1/20 0.49
PKM P14618 1/20 0.49
HDAC1 Q13547 1/20 0.49
TP53 P04637 2/20 0.48
UBE2I P63279 1/20 0.48
CACNA1B Q00975 1/20 0.48
APBA1 Q02410 1/20 0.48
SAE1 Q9UBE0 1/20 0.48
UBA2 Q9UBT2 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22972185 1.00 ALDH1A1 (0.58) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL22972399 0.92 HPGD (0.52) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL22972362 0.90 HPGD (0.66) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL22972401 0.85 HPGD (0.54) ALDH1A1KDM4EHPGDGAAHTT
SCHEMBL22972240 0.84 HPGD (0.57) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL22972410 0.84 GAA (0.52) HPGDGAA
SCHEMBL22972235 0.83 MAPT (0.55) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL30049303 0.83 DDR2 (0.54) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL29318681 0.83 DDR2 (0.54) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL24724231 0.83 KDR (0.54) HPGDGAADDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4010330-A1 QUINOLINE DERIVATIVES AS PROTEIN KINASE INHIBITORS B.C.I. Pharma (BE) 2022-06-15 EP disclosed