SCHEMBL29635376

SCHEMBL29635376

COc1nc(-c2ccc(C(F)(F)F)nc2)nc(F)c1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.43
CHEK1 O14757 1/20 0.38
TRPV3 Q8NET8 3/20 0.37
CASP3 P42574 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22042748 1.00 PDE10A (0.43) PDE10ACHEK1TRPV3CASP3KDM5B
SCHEMBL30969081 1.00 PDE10A (0.43) PDE10ACHEK1TRPV3CASP3KDM5B
SCHEMBL29635363 0.86 HDAC1 (0.41) HDAC1HDAC6HDAC5
SCHEMBL22042756 0.86 HDAC1 (0.36) PDE10ACHEK1HDAC1HDAC6HDAC5
SCHEMBL22042711 0.86 HDAC1 (0.41) HDAC1HDAC6HDAC5
SCHEMBL29635368 0.86 HDAC1 (0.36) PDE10ACHEK1HDAC1HDAC6HDAC5
SCHEMBL30969065 0.86 HDAC1 (0.41) HDAC1HDAC6HDAC5
SCHEMBL30421024 0.86 HDAC1 (0.36) PDE10ACHEK1HDAC1HDAC6HDAC5
SCHEMBL30151270 0.81 MAPT (0.43)
SCHEMBL22042751 0.81 S1PR1 (0.38) HDAC1HDAC6HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112739689-B Fluorine-containing pyrimidine compound and method for producing same 优迈特株式会社 2022-06-03 CN disclosed