SCHEMBL29638296

SCHEMBL29638296

COc1ccccc1/C=C1\C(=O)Nc2ccc(F)cc21

nearest known ligand 0.74

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.74
MEN1 O00255 2/20 0.73
KMT2A Q03164 2/20 0.73
CCNE1 P24864 2/20 0.67
CDK2 P24941 2/20 0.67
CCNE2 O96020 1/20 0.67
FLT3 P36888 7/20 0.65
MDM2 Q00987 4/20 0.62
RPS6KA3 P51812 1/20 0.59
KDR P35968 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14448964 0.86 MDM2 (0.68) NPC1MEN1KMT2ACCNE1CDK2
SCHEMBL5478629 0.86 MDM2 (0.68) NPC1MEN1KMT2ACCNE1CDK2
SCHEMBL5478628 0.86 MDM2 (0.68) NPC1MEN1KMT2ACCNE1CDK2
SCHEMBL5469888 0.86 MDM2 (0.74) NPC1MEN1KMT2AFLT3MDM2
SCHEMBL5469894 0.86 MDM2 (0.74) NPC1MEN1KMT2AFLT3MDM2
SCHEMBL7136252 0.86 NPC1 (0.72) NPC1MEN1KMT2ACCNE1CDK2
SCHEMBL5469692 0.85 NPC1 (1.00) NPC1CCNE1CDK2FLT3MDM2
SCHEMBL5469690 0.85 NPC1 (1.00) NPC1CCNE1CDK2FLT3MDM2
SCHEMBL16442345 0.85 NPC1 (1.00) NPC1CCNE1CDK2FLT3MDM2
SCHEMBL29367529 0.85 NPC1 (1.00) NPC1CCNE1CDK2FLT3MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111116452-B Indolone derivatives with alpha-glucosidase inhibitory activity as well as preparation method and application thereof 五邑大学 2022-05-03 CN disclosed