SCHEMBL7136252

SCHEMBL7136252

COc1ccccc1C=C1C(=O)Nc2ccc(I)cc21

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.72
MDM2 Q00987 3/20 0.58
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
MAPT P10636 4/20 0.53
APP P05067 2/20 0.53
CSNK1D P48730 3/20 0.51
CSNK1A1 P48729 2/20 0.51
CSNK1E P49674 2/20 0.51
GMNN O75496 2/20 0.51
LMNA P02545 2/20 0.51
TP53 P04637 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
HPGD P15428 2/20 0.51
MAPK1 P28482 2/20 0.51
CYP2C19 P33261 2/20 0.51
BLM P54132 2/20 0.51
PMP22 Q01453 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368659 0.89 NPC1 (0.57) NPC1MDM2MEN1KMT2AMAPT
SCHEMBL5369981 0.87 NPC1 (0.54) NPC1MDM2MEN1KMT2AMAPT
SCHEMBL29638296 0.86 NPC1 (0.74) NPC1MDM2MEN1KMT2ACCNE1
SCHEMBL5363455 0.86 MAPT (0.58) NPC1MDM2MEN1KMT2AMAPT
SCHEMBL5368424 0.85 MDM2 (0.61) NPC1MDM2MAPTAPPCSNK1D
SCHEMBL5358059 0.85 MDM2 (0.75) NPC1MDM2MAPTAPPCSNK1D
SCHEMBL5469894 0.85 MDM2 (0.74) NPC1MDM2MEN1KMT2AEGFR
SCHEMBL5469888 0.85 MDM2 (0.74) NPC1MDM2MEN1KMT2AEGFR
SCHEMBL5469690 0.84 NPC1 (1.00) NPC1MDM2MAPTCSNK1DCSNK1A1
SCHEMBL16442345 0.84 NPC1 (1.00) NPC1MDM2MAPTCSNK1DCSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed