SCHEMBL29638686

SCHEMBL29638686

Cc1ccc2c(Nc3cccc(C(F)(F)F)c3)nccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.52
ABCG2 Q9UNQ0 2/20 0.52
AURKA O14965 2/20 0.51
TSHR P16473 1/20 0.51
HTT P42858 1/20 0.51
PHGDH O43175 1/20 0.51
LMNA P02545 3/20 0.50
POLB P06746 1/20 0.50
APP P05067 1/20 0.50
LCK P06239 1/20 0.50
BRAF P15056 1/20 0.50
KDR P35968 1/20 0.50
TEK Q02763 1/20 0.50
MEN1 O00255 1/20 0.50
GMNN O75496 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TTR P02766 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30398394 0.84 ABCG2 (0.64) EGFRABCG2AURKATSHRHTT
SCHEMBL806052 0.84 ABCG2 (0.64) EGFRABCG2AURKATSHRHTT
SCHEMBL13686770 0.81 MAPK1 (0.56) EGFRABCG2HTTPOLBMEN1
SCHEMBL29638626 0.78 BRAF (0.58) EGFRABCG2TSHRHTTLMNA
SCHEMBL2261398 0.78 BRAF (0.58) EGFRABCG2AURKATSHRHTT
SCHEMBL2265817 0.78 BRAF (0.58) EGFRABCG2TSHRHTTLMNA
SCHEMBL30754777 0.78 LMNA (0.65) EGFRABCG2AURKATSHRHTT
SCHEMBL8373657 0.78 EGFR (0.76) EGFRABCG2TSHRHTTLMNA
SCHEMBL10215930 0.76 LMNA (0.64) EGFRABCG2AURKATSHRHTT
SCHEMBL10835262 0.75 LMNA (0.56) EGFRABCG2AURKATSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022089219-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2022-05-05 WO disclosed