SCHEMBL29640823

SCHEMBL29640823

O=C(O)c1ccccc1C1CN(c2nccc(-c3nccc(C#Cc4ccc5[nH]ncc5c4)n3)n2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 2/20 0.38
HCRTR1 O43613 6/20 0.37
HCRTR2 O43614 6/20 0.37
PDE10A Q9Y233 1/20 0.36
ROCK2 O75116 5/20 0.36
ROCK1 Q13464 2/20 0.36
PLK4 O00444 1/20 0.36
CHEK1 O14757 1/20 0.36
MAPK13 O15264 1/20 0.36
PDPK1 O15530 1/20 0.36
DAPK3 O43293 1/20 0.36
DYRK3 O43781 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
CHEK2 O96017 1/20 0.36
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29640799 0.88 ACACB (0.36) HAO1HCRTR1HCRTR2PDE10AROCK2
SCHEMBL29627898 0.87 HAO1 (0.39) HAO1HCRTR1HCRTR2PDE10AROCK2
Trifluoroacetic Acid SCHEMBL29640908 0.86 KDM1A (0.34) HAO1HCRTR1HCRTR2PDE10AROCK2
Trifluoroacetic Acid SCHEMBL29908226 0.85 ACACB (0.40) HAO1HCRTR1HCRTR2PDE10AROCK2
SCHEMBL29908258 0.83 ROCK2 (0.44) PDE10AROCK2ROCK1ACACBGRIN1
SCHEMBL29627921 0.81 ROCK2 (0.38) PDE10AROCK2ROCK1KDR
SCHEMBL29627883 0.81 ACACB (0.46) PDE10AROCK2ROCK1ACACBGRIN1
Trifluoroacetic Acid SCHEMBL29628004 0.81 ROCK2 (0.37) HAO1ROCK2ACACB
SCHEMBL29908262 0.80 ROCK2 (0.39) ROCK2ROCK1MAPK1GRIN1GRIN2B
SCHEMBL29627719 0.80 ROCK2 (0.53) ROCK2ROCK1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed