SCHEMBL29640905

SCHEMBL29640905

Oc1ccccc1N1CCN(c2nccc(-c3nccc(C#Cc4ccc5[nH]ncc5c4)n3)n2)CC1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
PIK3CA P42336 3/20 0.38
ROCK2 O75116 6/20 0.37
ROCK1 Q13464 3/20 0.37
TRPV1 Q8NER1 5/20 0.36
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
HTR1A P08908 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29908262 0.88 ROCK2 (0.39) GAAPIK3CAROCK2ROCK1GRIN1
SCHEMBL29627924 0.86 PIK3CA (0.40) PIK3CAROCK2ROCK1HTR1A
SCHEMBL29627719 0.84 ROCK2 (0.53) ROCK2ROCK1GRIN1GRIN2B
SCHEMBL29627883 0.83 ACACB (0.46) PIK3CAROCK2ROCK1GRIN1GRIN2B
SCHEMBL29627972 0.83 ROCK2 (0.38) ROCK2ROCK1GRIN1GRIN2BHTR1A
SCHEMBL29908257 0.83 GRIN2B (0.41) GAAPIK3CAROCK2ROCK1GRIN2B
SCHEMBL29908225 0.83 KCNH2 (0.43) ROCK2ROCK1TRPV1HTR1A
SCHEMBL29627894 0.82 ROCK2 (0.39) ROCK2ROCK1GRIN1GRIN2BHTR1A
SCHEMBL29627740 0.80 ROCK2 (0.44) ROCK2ROCK1
SCHEMBL29908258 0.80 ROCK2 (0.44) ROCK2ROCK1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed