SCHEMBL29644080

SCHEMBL29644080

Nc1ccc2[nH]nc(Br)c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 6/20 0.53
PDPK1 O15530 4/20 0.53
GSK3B P49841 1/20 0.51
AXL P30530 2/20 0.46
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
AURKA O14965 1/20 0.42
KDM4E B2RXH2 3/20 0.41
GAA P10253 2/20 0.41
MEN1 O00255 2/20 0.41
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
ROCK2 O75116 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
ROCK1 Q13464 1/20 0.41
HIF1A Q16665 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2467763 1.00 JAK2 (0.53) JAK2PDPK1GSK3BAXLHTR2A
SCHEMBL7571940 0.84 PDPK1 (0.53) JAK2PDPK1GSK3BAXLAURKA
SCHEMBL30860966 0.84 PDPK1 (0.53) JAK2PDPK1GSK3BAXLAURKA
SCHEMBL118573 0.81 JAK2 (0.64) JAK2PDPK1GSK3BAXLHTR2A
SCHEMBL30855645 0.79 PDPK1 (0.68) JAK2PDPK1GSK3BAXLHTR2A
SCHEMBL31584704 0.76 MAP2K4 (0.53) JAK2PDPK1KDM4EMAPTALDH1A1
SCHEMBL7571499 0.76 GSK3B (0.51) JAK2PDPK1GSK3BAXLHTR2A
SCHEMBL4004201 0.76 GSK3B (0.51) JAK2PDPK1GSK3BAXLHTR2A
SCHEMBL266855 0.76 GSK3B (0.56) JAK2PDPK1GSK3BAXLHTR2A
SCHEMBL759158 0.76 GSK3B (0.51) JAK2PDPK1GSK3BAXLHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3997081-A1 INDAZOLES AND AZAINDAZOLES AS LRRK2 INHIBITORS Escape Bio, Inc. (US) 2022-05-18 EP disclosed