SCHEMBL7571940

SCHEMBL7571940

Nc1ccc2c(Br)n[nH]c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 6/20 0.53
JAK2 O60674 3/20 0.53
AXL P30530 2/20 0.49
FGFR1 P11362 1/20 0.42
FGFR2 P21802 1/20 0.42
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.41
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
PKM P14618 1/20 0.41
HTT P42858 1/20 0.41
GSK3B P49841 2/20 0.40
PARP1 P09874 1/20 0.39
AURKA O14965 1/20 0.39
IMPDH2 P12268 1/20 0.38
PRKCI P41743 1/20 0.37
ROCK2 O75116 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30860966 1.00 PDPK1 (0.53) PDPK1JAK2AXLFGFR1FGFR2
SCHEMBL2467763 0.84 JAK2 (0.53) PDPK1JAK2AXLKDM4EMEN1
SCHEMBL29644080 0.84 JAK2 (0.53) PDPK1JAK2AXLKDM4EMEN1
SCHEMBL922069 0.81 PDPK1 (0.65) PDPK1JAK2AXLFGFR1FGFR2
SCHEMBL14755254 0.76 AXL (0.49) PDPK1JAK2AXLFGFR1FGFR2
SCHEMBL445902 0.76 FGFR1 (0.50) PDPK1JAK2AXLFGFR1FGFR2
SCHEMBL588513 0.76 AXL (0.50) PDPK1JAK2AXLFGFR1FGFR2
SCHEMBL15529807 0.76 GSK3B (0.48) PDPK1JAK2GSK3BPARP1ALDH1A1
SCHEMBL18764465 0.76 PDPK1 (0.44) PDPK1JAK2AXLFGFR1FGFR2
SCHEMBL2926172 0.76 AXL (0.49) PDPK1JAK2AXLFGFR1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904769-B1 Keratin fibre dye compositions containing Indazole amine derivatives and dyeing method OREAL (FR) 2002-09-25 EP claimed
WO-2025129167-A1 INHIBITORS OF THE SURFACE EXPRESSION OF THE VOLTAGE-GATED SODIUM ION CHANNEL 1.7 (NAV1.7) AND THEIR THERAPEUTIC USES THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2025-06-19 WO disclosed
US-20240174647-A1 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. 2024-05-30 US disclosed
WO-2024073073-A2 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. (US) 2024-04-04 WO disclosed
US-6027538-A OXIDATION DYEING OF KERATINOUS FIBERS CONTAINING AT LEAST ONE COUPLER SELECTED FROM INDAZOLEAMINE DERIVATIVES AND AT LEAST ONE OXIDATION BASE; POWERFUL, NOT VERY SELECTIVE HAIR DYES WHICH ARE CAPABLE OF GENERATING INTENSE COLOR L'OREAL S.A. (FR) 2000-02-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240174647-A1 KINASE MODULATORS AND METHODS OF USE THEREOF LRRK2, MAP3K20, MAP3K5 PDPK1 42/4885JAK2 352/4885AXL 624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.