SCHEMBL29644385

SCHEMBL29644385

CCOC(=O)CC(CCc1cn(C)nn1)c1cccc2c1CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.38
NQO1 P15559 1/20 0.37
ADORA1 P30542 1/20 0.36
UCHL1 P09936 1/20 0.36
MAP3K5 Q99683 3/20 0.35
ESR2 Q92731 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MAPK1 P28482 1/20 0.35
NR1H2 P55055 1/20 0.35
NAMPT P43490 1/20 0.35
C5AR1 P21730 2/20 0.34
ACACB O00763 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
P2RX3 P56373 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
ABHD6 Q9BV23 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28739021 1.00 SCN9A (0.38) SCN9ANQO1ADORA1UCHL1MAP3K5
SCHEMBL28739042 0.92 NQO1 (0.46) SCN9ANQO1ADORA1UCHL1MAP3K5
SCHEMBL29644414 0.92 NQO1 (0.46) SCN9ANQO1ADORA1UCHL1MAP3K5
SCHEMBL25299079 0.84 ADORA1 (0.43) SCN9AADORA1UCHL1ESR2TMEM97
SCHEMBL31057139 0.84 ADORA1 (0.43) SCN9AADORA1UCHL1ESR2TMEM97
SCHEMBL25299080 0.84 ADORA1 (0.43) SCN9AADORA1UCHL1ESR2TMEM97
SCHEMBL28739147 0.84 LMNA (0.37) NAMPTKMT2APOLBMAPT
SCHEMBL29201185 0.83 NQO1 (0.55) SCN9ANQO1UCHL1ESR2
SCHEMBL25259759 0.80 ADORA1 (0.46) SCN9AADORA1UCHL1MAP3K5ESR2
SCHEMBL25300998 0.80 ADORA1 (0.46) SCN9AADORA1UCHL1MAP3K5ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed
CN-114507181-A Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-05-17 CN disclosed