SCHEMBL29644465

SCHEMBL29644465

CCOC(=O)CC(c1ccccc1)c1cccc2c1CCN(Cc1ccccc1)C2

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 13/20 0.50
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
ADORA1 P30542 1/20 0.47
NPC1 O15118 1/20 0.43
TNF P01375 1/20 0.43
RAB9A P51151 1/20 0.43
NOD2 Q9HC29 1/20 0.43
NOD1 Q9Y239 1/20 0.43
ABCB1 P08183 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28739068 1.00 ACACB (0.50) ACACBMEN1KMT2ALMNAMAPT
SCHEMBL28739144 0.93 ACACB (0.48) ACACBMEN1KMT2ALMNAMAPT
SCHEMBL29644413 0.93 ACACB (0.48) ACACBMEN1KMT2ALMNAMAPT
SCHEMBL28739024 0.90 ACACB (0.46) ACACBMEN1KMT2ALMNAMAPT
SCHEMBL29644350 0.90 ACACB (0.46) ACACBMEN1KMT2ALMNAMAPT
SCHEMBL28739185 0.86 ACACB (0.53) ACACBMEN1KMT2AADORA1
SCHEMBL29644415 0.86 ACACB (0.53) ACACBMEN1KMT2AADORA1
SCHEMBL28739132 0.82 KEAP1 (0.44) MEN1KMT2ALMNA
SCHEMBL29644302 0.82 KEAP1 (0.44) MEN1KMT2ALMNA
SCHEMBL28738983 0.81 FFAR1 (0.51) ACACBTNFNOD2NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed
CN-114507181-A Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-05-17 CN disclosed