SCHEMBL29646014

SCHEMBL29646014

CC(C)n1cc(-c2nc3c4cccc(F)c4nc(N[C@@H]4CN(C(=O)OCc5ccccc5)CCNC4=O)n3n2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
PARP1 P09874 5/20 0.33
TRPC3 Q13507 1/20 0.33
TRPC7 Q9HCX4 1/20 0.33
USP30 Q70CQ3 1/20 0.33
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
GABRA5 P31644 1/20 0.32
JAK2 O60674 3/20 0.32
JAK1 P23458 3/20 0.32
TYK2 P29597 2/20 0.32
JAK3 P52333 2/20 0.32
LCK P06239 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22988001 1.00 NR1H2 (0.33) NR1H2NR1H3PARP1TRPC3TRPC7
SCHEMBL22987658 0.93 NR1H2 (0.37) NR1H2NR1H3PARP1TRPC3TRPC7
SCHEMBL25118878 0.93 NR1H2 (0.37) NR1H2NR1H3PARP1TRPC3TRPC7
SCHEMBL22988171 0.93 ADORA3 (0.35) PARP1TRPC3TRPC7USP30GABRA5
SCHEMBL22988242 0.93 USP30 (0.33) NR1H2NR1H3PARP1USP30TP53
SCHEMBL22987728 0.93 USP30 (0.33) NR1H2NR1H3PARP1USP30TP53
SCHEMBL22987791 0.93 TRPC3 (0.33) NR1H2NR1H3PARP1TRPC3TRPC7
SCHEMBL25118615 0.92 JAK2 (0.34) PARP1TRPC3TRPC7USP30TP53
SCHEMBL25118622 0.92 USP30 (0.32) NR1H2NR1H3PARP1USP30TP53
SCHEMBL22988270 0.91 USP30 (0.34) NR1H2NR1H3PARP1TRPC3TRPC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed