SCHEMBL29646407

SCHEMBL29646407

COc1ccc(-c2nc3c4cccc(SC)c4nc(Cl)n3n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
POLB P06746 1/20 0.48
ADORA3 P0DMS8 11/20 0.45
ADORA1 P30542 5/20 0.43
ADORA2A P29274 4/20 0.43
MAPT P10636 3/20 0.42
THRB P10828 1/20 0.42
XDH P47989 1/20 0.42
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
LIPE Q05469 1/20 0.40
RAB9A P51151 2/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979525 1.00 KDM4E (0.48) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL30393698 0.88 ADORA3 (0.48) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL22988213 0.88 ADORA3 (0.48) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL22987710 0.88 KDM4E (0.46) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL30393525 0.88 KDM4E (0.46) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL22988185 0.87 ADORA3 (0.56) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL22988147 0.86 KDM4E (0.52) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL22987552 0.85 KDM4E (0.51) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL22987426 0.85 KDM4E (0.51) KDM4EALDH1A1POLBADORA3ADORA1
SCHEMBL22987462 0.84 KDM4E (0.50) KDM4EALDH1A1POLBADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-B [1,2,4] Triazolo [1,5-C ] quinazolin-5-amine 拜耳股份有限公司 2024-09-10 CN disclosed
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN disclosed