SCHEMBL29646465

SCHEMBL29646465

COc1cccc(-c2nc3c4ccccc4[nH]c(=O)n3n2)c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.77
ALDH1A1 P00352 2/20 0.77
POLB P06746 1/20 0.77
GABRP O00591 1/20 0.70
GABRD O14764 1/20 0.70
GABRA1 P14867 1/20 0.70
GABRB1 P18505 1/20 0.70
GABRG2 P18507 1/20 0.70
GABRB3 P28472 1/20 0.70
GABRA5 P31644 1/20 0.70
GABRA3 P34903 1/20 0.70
GABRA2 P47869 1/20 0.70
GABRB2 P47870 1/20 0.70
GABRA4 P48169 1/20 0.70
GABRE P78334 1/20 0.70
GABRA6 Q16445 1/20 0.70
GABRG1 Q8N1C3 1/20 0.70
GABRG3 Q99928 1/20 0.70
GABRQ Q9UN88 1/20 0.70
HSD17B10 Q99714 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979083 1.00 KDM4E (0.77) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL22987849 0.88 KDM4E (0.62) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL22987773 0.88 KDM4E (0.62) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL29646388 0.87 KDM4E (1.00) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL22979094 0.87 KDM4E (1.00) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL22987929 0.87 KDM4E (0.61) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL22987775 0.87 KDM4E (0.61) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL22987526 0.86 GABRP (0.65) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL22979129 0.85 TP53 (0.76) KDM4EALDH1A1POLBGABRPGABRD
SCHEMBL29646398 0.85 TP53 (0.76) KDM4EALDH1A1POLBGABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-B [1,2,4] Triazolo [1,5-C ] quinazolin-5-amine 拜耳股份有限公司 2024-09-10 CN disclosed
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN disclosed