SCHEMBL29646480

SCHEMBL29646480

COc1ccc(-c2nc3c4cccc(Br)c4nc(N[C@@H]4CN(C(=O)OCc5ccccc5)CCNC4=O)n3n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.40
MMP9 P14780 5/20 0.40
MMP1 P03956 4/20 0.40
MMP3 P08254 4/20 0.40
MMP7 P09237 3/20 0.40
MMP13 P45452 2/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
MAPT P10636 3/20 0.38
THRB P10828 1/20 0.38
ADAM17 P78536 1/20 0.38
ADAM9 Q13443 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
PARP1 P09874 1/20 0.36
MMP2 P08253 1/20 0.36
MMP8 P22894 1/20 0.36
BCL9 O00512 1/20 0.36
CTNNB1 P35222 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22988011 1.00 ADORA3 (0.40) ADORA3MMP9MMP1MMP3MMP7
SCHEMBL22987600 1.00 ADORA3 (0.40) ADORA3MMP9MMP1MMP3MMP7
SCHEMBL22988314 0.93 ADORA3 (0.40) ADORA3MMP9MMP1MMP3MMP7
SCHEMBL22987917 0.93 MAPT (0.42) ADORA3MMP9MMP1MMP3MMP7
SCHEMBL30393181 0.93 ADORA3 (0.40) ADORA3MMP9MMP1MMP3MMP7
SCHEMBL22987627 0.92 ADORA3 (0.40) ADORA3MMP9MMP1MMP3MMP7
SCHEMBL25118867 0.92 ADORA3 (0.40) ADORA3MMP9MMP1MMP3MMP7
SCHEMBL22988108 0.92 TRPC3 (0.39) ADORA3ADORA2AADORA1MAPTKDM1A
SCHEMBL22987799 0.92 TRPC3 (0.39) ADORA3ADORA2AADORA1MAPTKDM1A
SCHEMBL22987722 0.92 TRPC3 (0.39) ADORA3ADORA2AADORA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN disclosed