SCHEMBL29648738

SCHEMBL29648738

O=C1NCCCC[C@H]1Nc1nc2c(C(F)(F)F)cccc2c2nc(-c3ccc(Cl)cc3OC(F)(F)F)nn12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.34
TACR2 P21452 8/20 0.34
ADORA2A P29274 6/20 0.33
ADORA1 P30542 6/20 0.33
KCNH2 Q12809 4/20 0.33
CYP3A4 P08684 3/20 0.33
ADORA3 P0DMS8 2/20 0.33
ADORA2B P29275 1/20 0.33
CYP2C19 P33261 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NR1I2 O75469 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
HTR1A P08908 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
CNR1 P21554 1/20 0.33
GLRA1 P23415 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979089 1.00 TACR1 (0.34) TACR1TACR2ADORA2AADORA1KCNH2
SCHEMBL29648590 0.92 ADORA2A (0.34) TACR1TACR2ADORA2AADORA1KCNH2
SCHEMBL22988429 0.92 ADORA2A (0.34) TACR1TACR2ADORA2AADORA1KCNH2
SCHEMBL29648704 0.91 TACR1 (0.32) TACR1TACR2NPC1RAB9A
SCHEMBL22978985 0.91 TACR1 (0.32) TACR1TACR2NPC1RAB9A
SCHEMBL22980169 0.91 TACR1 (0.32) TACR1TACR2NPC1RAB9A
SCHEMBL29648710 0.91 TACR1 (0.32) TACR1TACR2NPC1RAB9A
SCHEMBL22988434 0.90 PLAT (0.30)
SCHEMBL29645872 0.90 PLAT (0.30)
SCHEMBL22988022 0.88 MKNK1 (0.36) TACR1TACR2ADORA2AADORA1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-B [1,2,4] Triazolo [1,5-C ] quinazolin-5-amine 拜耳股份有限公司 2024-09-10 CN claimed
EP-4013508-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES Bayer Aktiengesellschaft (DE) 2022-06-22 EP claimed