SCHEMBL29654023

SCHEMBL29654023

NC(=O)c1snc2cccnc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 2/20 0.51
PARP1 P09874 1/20 0.45
IKBKB O14920 2/20 0.44
CHUK O15111 1/20 0.44
KDM4E B2RXH2 3/20 0.41
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
HPGD P15428 2/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MKNK2 Q9HBH9 3/20 0.35
MKNK1 Q9BUB5 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PLK4 O00444 1/20 0.35
MAP4K4 O95819 1/20 0.35
EGFR P00533 1/20 0.35
ROS1 P08922 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23495057 0.84 KDM4E (0.40) LIMK1PARP1KDM4EJAK2JAK1
SCHEMBL23514475 0.79 KDM4E (0.46) KDM4EJAK2JAK1TYK2JAK3
SCHEMBL4603472 0.73 LIMK1 (0.44) LIMK1PARP1IKBKBCHUKL3MBTL1
SCHEMBL4072413 0.72 PRMT5 (0.42) LIMK1KDM4EHTTSMN1; SMN2L3MBTL1
Hydrochloric Acid SCHEMBL4603416 0.71 LIMK1 (0.43) LIMK1PARP1IKBKBCHUKKDM4E
SCHEMBL21139553 0.70 KDM4E (0.39) KDM4EHPGDHTTSMN1; SMN2L3MBTL1
SCHEMBL19554538 0.69 LIMK1 (0.51) LIMK1PARP1IKBKBCHUKKDM4E
SCHEMBL30001410 0.69 PARP1 (0.53) LIMK1PARP1IKBKBCHUKKDM4E
SCHEMBL23495082 0.68 KDM4E (0.38) KDM4EHTTSMN1; SMN2L3MBTL1EGFR
SCHEMBL4069439 0.68 HSP90AA1 (0.43) KDM4EHTTSMN1; SMN2L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110494434-B Pyrazolophenyl compounds, compositions thereof, and methods of use thereof 豪夫迈·罗氏有限公司 2022-05-24 CN disclosed