SCHEMBL29654089

SCHEMBL29654089

NC(=S)c1csc(Nc2cccc(Cl)c2)n1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.70
MAPT P10636 9/20 0.56
GAA P10253 4/20 0.56
CYP1A2 P05177 2/20 0.53
CYP1A1 P04798 1/20 0.53
CYP1B1 Q16678 1/20 0.53
MEN1 O00255 7/20 0.52
KMT2A Q03164 7/20 0.52
ALDH1A1 P00352 5/20 0.52
SMN1; SMN2 Q16637 4/20 0.51
LMNA P02545 3/20 0.51
ALOX12 P18054 1/20 0.51
HTT P42858 1/20 0.51
ALOX5 P09917 1/20 0.48
CFTR P13569 2/20 0.47
KDM4E B2RXH2 3/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
GLA P06280 1/20 0.46
NPC1 O15118 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28716317 1.00 KDM1A (0.70) KDM1AMAPTGAACYP1A2CYP1A1
SCHEMBL29654005 0.86 KDM1A (0.78) KDM1AMAPTGAACYP1A2CYP1A1
SCHEMBL28707161 0.86 KDM1A (0.78) KDM1AMAPTGAACYP1A2CYP1A1
SCHEMBL28716330 0.85 ALOX5 (0.52) KDM1AMAPTGAACYP1A2CYP1A1
SCHEMBL28713943 0.83 CYP1A2 (0.53) KDM1AMAPTCYP1A2CYP1A1CYP1B1
SCHEMBL29654077 0.83 CYP1A2 (0.53) KDM1AMAPTCYP1A2CYP1A1CYP1B1
SCHEMBL2870272 0.83 KDM1A (0.78) KDM1AMAPTGAACYP1A2CYP1A1
SCHEMBL28717687 0.82 KDM1A (0.67) KDM1AMAPTGAACYP1A2CYP1A1
SCHEMBL2880884 0.77 KDM1A (0.72) KDM1AMAPTGAACYP1A2CYP1A1
SCHEMBL23553978 0.74 CFTR (0.77) KDM1AMAPTCYP1A2CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-B N-aryl- [2,4 '-dithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2023-09-05 CN disclosed
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed