SCHEMBL29654752

SCHEMBL29654752

COC(=O)c1cc(I)c(-c2ccc(F)cc2F)cc1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 7/20 0.56
ALPL P05186 1/20 0.45
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 5/20 0.42
MAPT P10636 4/20 0.42
HSD17B10 Q99714 3/20 0.42
HPGD P15428 3/20 0.42
GAA P10253 2/20 0.42
GLA P06280 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
ATM Q13315 1/20 0.42
ABL1 P00519 1/20 0.41
TTR P02766 1/20 0.41
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
IKBKB O14920 1/20 0.39
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23540616 1.00 CFTR (0.56) CFTRALPLKDM4EALDH1A1MAPT
SCHEMBL23556347 0.85 ALPL (0.46) CFTRALPLKDM4EALDH1A1MAPT
SCHEMBL29476152 0.85 SLC6A4 (0.56) CFTRKDM4EALDH1A1MAPTHSD17B10
SCHEMBL23540082 0.85 SLC6A4 (0.56) CFTRKDM4EALDH1A1MAPTHSD17B10
SCHEMBL23539893 0.84 ABL1 (0.48) CFTRALPLKDM4EALDH1A1MAPT
SCHEMBL29476388 0.84 ABL1 (0.48) CFTRALPLKDM4EALDH1A1MAPT
SCHEMBL23539858 0.83 TTR (0.55) CFTRKDM4EALDH1A1MAPTHSD17B10
SCHEMBL29476378 0.82 CFTR (0.56) CFTRALPLKDM4EALDH1A1MAPT
SCHEMBL23539751 0.82 CFTR (0.56) CFTRALPLKDM4EALDH1A1MAPT
SCHEMBL23539577 0.81 ALPL (0.43) CFTRALPLKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022133345-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. (US) 2022-06-23 WO disclosed