SCHEMBL29655115

SCHEMBL29655115

Nc1ccc(-c2ccccc2F)cc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
PTPRC P08575 1/20 0.52
PTPN1 P18031 1/20 0.52
MAP4K4 O95819 1/20 0.50
FEN1 P39748 5/20 0.49
ALOX5AP P20292 4/20 0.49
ACMSD Q8TDX5 1/20 0.46
TRPA1 O75762 1/20 0.45
PDK2 Q15119 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ADORA1 P30542 1/20 0.42
PGR P06401 1/20 0.42
TNKS O95271 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5952352 1.00 BACE1 (0.53) BACE1MEN1KMT2ATDP1PTPRC
SCHEMBL29655190 1.00 BACE1 (0.53) BACE1MEN1KMT2ATDP1PTPRC
Ammonia Solution, Strong SCHEMBL5953223 0.98 BACE1 (0.51) BACE1MEN1KMT2ATDP1PTPRC
SCHEMBL15250336 0.88 BACE1 (0.53) BACE1TDP1PTPRCPTPN1MAP4K4
SCHEMBL29655217 0.84 MEN1 (0.48) BACE1MEN1KMT2ATDP1PTPRC
SCHEMBL23040370 0.82 TNKS (0.49) BACE1TDP1PTPRCPTPN1MAP4K4
SCHEMBL5843391 0.82 ALOX15 (0.57) BACE1MEN1KMT2APTPRCPTPN1
SCHEMBL29878768 0.82 ALOX15 (0.57) BACE1MEN1KMT2APTPRCPTPN1
SCHEMBL5556308 0.80 MEN1 (0.59) MEN1KMT2ATDP1FEN1ALOX5AP
SCHEMBL28602582 0.80 BACE1 (0.46) BACE1PTPRCPTPN1MAP4K4FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843874-B Phthalazine derivatives useful as inhibitors of PARP1, PARP2 and/or tubulin for the treatment of cancer 加利福尼亚大学董事会 2022-05-27 CN disclosed