SCHEMBL29655475

SCHEMBL29655475

CC(=O)Nc1cccc(Nc2nc(Cl)ncc2Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.57
CTSC P53634 1/20 0.57
CCNT1 O60563 1/20 0.57
CCNK O75909 1/20 0.57
CYP3A4 P08684 1/20 0.57
CCND3 P30281 1/20 0.57
CDK9 P50750 1/20 0.57
CDK6 Q00534 1/20 0.57
ABCG2 Q9UNQ0 3/20 0.52
MAP3K5 Q99683 1/20 0.52
EGFR P00533 8/20 0.52
AURKA O14965 1/20 0.51
AURKB Q96GD4 1/20 0.51
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
MAPT P10636 1/20 0.49
MAPK1 P28482 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28782963 1.00 CTSL (0.57) CTSLCTSCCCNT1CCNKCYP3A4
SCHEMBL264837 0.88 EGFR (0.54) CTSLCTSCCCNT1CCNKCYP3A4
SCHEMBL1036047 0.87 EGFR (0.53) CCNT1CDK9ABCG2MAP3K5EGFR
SCHEMBL30395760 0.86 POLB (0.57) CTSCCYP3A4EGFRAURKAALDH1A1
SCHEMBL29019906 0.86 POLB (0.57) CTSCCYP3A4EGFRAURKAALDH1A1
SCHEMBL24842760 0.85 CTSC (0.63) CTSLCTSCCCNT1CCNKCYP3A4
SCHEMBL29816657 0.85 CTSC (0.63) CTSLCTSCCCNT1CCNKCYP3A4
SCHEMBL17197435 0.84 EGFR (0.52) ABCG2MAP3K5EGFR
SCHEMBL9945478 0.84 BTK (0.67) EGFR
SCHEMBL4180112 0.83 SYK (0.57) CTSLCTSCCCNT1CCNKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121248582-B CDK12/PARP double-target inhibitor and preparation method and application thereof SOUTH CHINA UNIVERSITY OF TECHNOLOGY (CN) 2026-05-26 CN disclosed
CN-114621206-B 5-substituted pyrimidine diamine derivative and preparation method and application thereof 安徽医科大学 2023-11-24 CN disclosed
CN-111620852-B 5-chloro-pyrimidine-2, 4-diamine compound, and preparation method and application thereof 镇江植生源农业科技有限公司 2023-05-09 CN disclosed
CN-114621206-A 5-substituted pyrimidinediamine derivative and preparation method and application thereof 安徽医科大学 2022-06-14 CN disclosed