SCHEMBL29658372

SCHEMBL29658372

Nc1cc(C(=O)NCCN2CCCC2)cc(C(F)(F)F)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.63
KMT2A Q03164 1/20 0.63
EPHX2 P34913 4/20 0.59
CD274 Q9NZQ7 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.50
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
ALDH1A1 P00352 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28735422 1.00 MEN1 (0.63) MEN1KMT2AEPHX2CD274SMN1; SMN2
SCHEMBL29658388 0.99 MEN1 (0.62) MEN1KMT2AEPHX2CD274SMN1; SMN2
SCHEMBL28735420 0.99 MEN1 (0.62) MEN1KMT2AEPHX2CD274SMN1; SMN2
SCHEMBL28735408 0.97 MEN1 (0.60) MEN1KMT2AEPHX2CD274SMN1; SMN2
SCHEMBL29658312 0.97 MEN1 (0.60) MEN1KMT2AEPHX2CD274SMN1; SMN2
SCHEMBL2967384 0.89 CD274 (0.66) EPHX2CD274ALDH1A1CYP1A2CYP2D6
SCHEMBL29658344 0.89 CD274 (0.66) EPHX2CD274ALDH1A1CYP1A2CYP2D6
SCHEMBL28735410 0.88 MEN1 (0.49) MEN1KMT2AEPHX2CD274CHRNB2
SCHEMBL28735456 0.88 MEN1 (0.49) MEN1KMT2AEPHX2CD274CHRNB2
SCHEMBL28735345 0.85 MEN1 (0.45) MEN1KMT2AEPHX2CD274ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478366-A Pyridone derivative and application thereof in medicine 海思科医药集团股份有限公司 2022-05-13 CN disclosed