SCHEMBL2966032

SCHEMBL2966032

Brc1ncnc2oc(-c3ccccc3)c(-c3ccccc3)c12

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TNK2 Q07912 1/20 0.68
ALDH1A1 P00352 2/20 0.57
HPGD P15428 2/20 0.57
TSHR P16473 1/20 0.57
HSD17B10 Q99714 1/20 0.57
AURKA O14965 11/20 0.56
CHEK1 O14757 3/20 0.56
MAP2K1 Q02750 1/20 0.56
EGFR P00533 2/20 0.54
KDM4E B2RXH2 1/20 0.54
UBE2N P61088 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
RAD52 P43351 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13271835 0.81 TNK2 (0.68) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL735560 0.81 TNK2 (0.68) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL2965887 0.81 TNK2 (1.00) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL2976986 0.81 TNK2 (0.68) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL1787179 0.80 TNK2 (0.58) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL2966671 0.77 ALDH1A1 (0.64) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL3561541 0.74 TNK2 (0.51) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL13632594 0.74 AURKA (0.81) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL2977130 0.74 TNK2 (0.58) TNK2ALDH1A1HPGDTSHRHSD17B10
SCHEMBL6848486 0.74 TNK2 (0.58) TNK2ALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7776867-B2 Furanopyrimidines AMGEN INC. (US) 2010-08-17 US disclosed
US-7776867-B2 Furanopyrimidines AMGEN INC. (US) 2010-08-17 US disclosed
US-7776867-B2 Furanopyrimidines AMGEN INC. (US) 2010-08-17 US disclosed
EP-1768986-A2 FURANOPYRIMIDINES Amgen Inc. (US) 2007-04-04 EP disclosed
US-20060040961-A1 Furanopyrimidines AMGEN INC. 2006-02-23 US disclosed
WO-2006004658-A2 FURANOPYRIMIDINES AMGEN INC. (US) 2006-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060040961-A1 Furanopyrimidines TYMS, IDO1, NFATC1 TNK2 1075/4885ALDH1A1 159/4885HPGD 1536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.