SCHEMBL29660550

SCHEMBL29660550

Fc1cnc2[nH]cc(Br)c2c1F

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.38
AXL P30530 1/20 0.35
HTR1A P08908 1/20 0.31
HTR7 P34969 1/20 0.31
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26965747 1.00 MAPK1 (0.38) MAPK1AXLHTR1AHTR7HTR6
SCHEMBL20575800 0.81 DAO (0.41) MAPK1AXL
SCHEMBL21632480 0.81 MAPK1 (0.36) MAPK1AXLHTR1AHTR7HTR6
SCHEMBL30321255 0.81 DAO (0.41) MAPK1AXL
SCHEMBL1468379 0.77 GSK3B (0.37)
SCHEMBL21632471 0.73 AXL (0.47) MAPK1AXL
SCHEMBL29722097 0.73 AXL (0.47) MAPK1AXL
SCHEMBL21632550 0.73 AXL (0.41) AXL
SCHEMBL1564880 0.72 DAO (0.35) MAPK1AXL
SCHEMBL24682764 0.70 TRPA1 (0.38) MAPK1AXLHTR1AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4247812-A1 SUBSTITUTED PYRROLO [2, 3-B] PYRIDINE AND PYRAZOLO [3, 4-B] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS Fochon Biosciences, Ltd. (CN) 2023-09-27 EP disclosed
CN-116568686-A Substituted pyrrolo [2,3-b ] pyridine and pyrazolo [3,4-b ] pyridine derivatives as protein kinase inhibitors 重庆复尚源创医药技术有限公司 2023-08-08 CN disclosed
WO-2022105746-A1 SUBSTITUTED PYRROLO [2, 3-b] PYRIDINE AND PYRAZOLO [3, 4-b] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS FOCHON PHARMACEUTICALS, LTD. (CN) 2022-05-27 WO disclosed