SCHEMBL29672802

SCHEMBL29672802

COc1cccc(-c2nnn[nH]2)n1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BTK Q06187 3/20 0.56
IDH1 O75874 1/20 0.36
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
APLNR P35414 3/20 0.34
KDR P35968 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA3 P34903 1/20 0.34
CNR1 P21554 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
TGFBR1 P36897 2/20 0.33
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15886669 1.00 BTK (0.56) BTKIDH1DDB1CRBNAPLNR
SCHEMBL12075530 0.82 MEN1 (0.36) BTK
SCHEMBL12598648 0.80 CCR1 (0.37) BTK
SCHEMBL12598652 0.80 CCR1 (0.37) BTK
SCHEMBL6982246 0.77 CCR1 (0.54) BTKTGFBR1
SCHEMBL3155981 0.75 BTK (0.61) BTKIDH1DDB1CRBNAPLNR
SCHEMBL30433661 0.74 ASIC3 (0.46) IDH1
SCHEMBL20557572 0.74 ASIC3 (0.46) IDH1
SCHEMBL19919698 0.73 BTK (0.31) BTKTGFBR1
SCHEMBL732877 0.73 BTK (0.34) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114585625-A Triazolopyrimidines as A2A/A2B inhibitors 因赛特公司 2022-06-03 CN disclosed