SCHEMBL29673283

SCHEMBL29673283

CC(C)(C)OC(=O)NCc1cc2nc(-c3cccc(N4CCC4)n3)ccc2cn1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 3/20 0.40
SKP1 P63208 3/20 0.40
SKP2 Q13309 3/20 0.40
CNR1 P21554 8/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
ACACB O00763 3/20 0.36
ACACA Q13085 3/20 0.36
IRAK1 P51617 1/20 0.36
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29070067 1.00 CKS1B (0.40) CKS1BSKP1SKP2CNR1L3MBTL1
SCHEMBL23731714 0.88 BRD4 (0.40) CKS1BSKP1SKP2ACACBACACA
SCHEMBL30103140 0.88 BRD4 (0.40) CKS1BSKP1SKP2ACACBACACA
SCHEMBL31396177 0.88 CKS1B (0.36) CKS1BSKP1SKP2ACACBACACA
SCHEMBL31401524 0.87 CKS1B (0.34) CKS1BSKP1SKP2L3MBTL1ACACB
SCHEMBL23706015 0.87 L3MBTL1 (0.41) CKS1BSKP1SKP2L3MBTL1ACACB
SCHEMBL26970021 0.86 CNR1 (0.43) CNR1ADORA2AADORA1PIM1PIM2
SCHEMBL31401234 0.86 EGLN1 (0.35) CKS1BSKP1SKP2ACACBACACA
SCHEMBL30689837 0.85 CNR1 (0.38) CNR1PIM1PIM2
SCHEMBL31396029 0.85 RET (0.38) CKS1BSKP1SKP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4244213-A1 COMPOUNDS AND USES THEREOF Foghorn Therapeutics Inc. (US) 2023-09-20 EP disclosed
WO-2022103899-A1 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. (US) 2022-05-19 WO disclosed