SCHEMBL29675604

SCHEMBL29675604

CCC(=O)N[C@H](C)c1ccnc(N2CCOCC2)c1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.52
MAPK1 P28482 3/20 0.46
RAF1 P04049 3/20 0.44
BRAF P15056 3/20 0.44
ACACB O00763 7/20 0.44
SHMT2 P34897 1/20 0.43
LRRK2 Q5S007 1/20 0.42
TRPV3 Q8NET8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29676386 0.87 HRH4 (0.44) MAPK1ACACBLRRK2
SCHEMBL29676029 0.86 PIK3CA (0.50) PIK3CAMAPK1RAF1BRAFSHMT2
SCHEMBL29675876 0.82 ACACB (0.49) MAPK1ACACB
SCHEMBL29675982 0.82 ACACB (0.49) MAPK1ACACB
SCHEMBL29675718 0.78 ACACB (0.52) MAPK1ACACB
SCHEMBL29676091 0.78 ACACB (0.52) MAPK1ACACB
SCHEMBL18931264 0.77 PIK3CA (0.51) PIK3CALRRK2TRPV3
SCHEMBL29676120 0.77 ACACB (0.48) ACACB
SCHEMBL1911474 0.77 PIK3CA (0.54) PIK3CARAF1BRAFLRRK2
SCHEMBL18704867 0.76 PIK3CA (0.52) PIK3CALRRK2TRPV3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617166-B Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-05-17 CN claimed