SCHEMBL2967589

SCHEMBL2967589

NC1CCC(c2ccccc2)c2ccccc21

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.62
SLC6A4 P31645 1/20 0.62
SLC6A3 Q01959 1/20 0.62
SIGMAR1 Q99720 2/20 0.46
KDM1A O60341 1/20 0.45
MAOB P27338 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5815434 1.00 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
SCHEMBL7330612 1.00 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
SCHEMBL5815432 1.00 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
SCHEMBL7330624 1.00 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
Hydrochloric Acid SCHEMBL11694448 0.98 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
Hydrochloric Acid SCHEMBL11694454 0.98 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
Hydrochloric Acid SCHEMBL11695457 0.98 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
Hydrochloric Acid SCHEMBL11695440 0.98 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3SIGMAR1KDM1A
SCHEMBL4367085 0.85 SLC6A2 (0.69) SLC6A2SLC6A4SLC6A3
SCHEMBL6924410 0.82 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3KDM1AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 80 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020035105-A1 Composition and method combining an antidepressant with an NMDA receptor antagonist, for treating neuropathic pain ENDO PHARMACEUTICALS INC. 2002-03-21 US claimed
EP-0980247-A1 COMPOSITION AND METHOD COMBINING AN ANTIDEPRESSANT WITH AN NMDA RECEPTOR ANTAGONIST, FOR TREATING NEUROPATHIC PAIN Algos Pharmaceutical Corporation (US) 2000-02-23 EP claimed
WO-1998050044-A1 COMPOSITION AND METHOD COMBINING AN ANTIDEPRESSANT WITH AN NMDA RECEPTOR ANTAGONIST, FOR TREATING NEUROPATHIC PAIN ALGOS PHARMACEUTICAL CORPORATION (US) 1998-11-12 WO claimed
US-4045488-A ANTIDEPRESSANTS OR PSYCHOMOTOR STIMULANTS PFIZER INC. (US) 1977-08-30 US claimed
US-4029731-A TREATING DEPRESSION PFIZER INC. (US) 1977-06-14 US claimed
JP-7173056-A None JP disclosed
JP-7173056-A None JP disclosed
EP-3712128-A1 PHOTOCHEMICAL INTERMOLECULAR AMINATION METHOD Fundació Institut Català d'Investigació Química (ICIQ) (ES) 2020-09-23 EP disclosed
EP-1542961-B1 TRANS 4-(3,4-DICHLOROPHENYL)-1,2,3,4-TETRAHYDRO-1-NAPTHALENAMINE FOR USE IN TREATMENT OF CNS DISORDERS SEPRACOR INC (US) 2013-09-11 EP disclosed
US-7772437-B2 Process of making sertraline form II HETERO DRUGS LIMITED (IN) 2010-08-10 US disclosed
US-7772438-B2 Process of making sertraline form I HETERO DRUGS LIMITED (IN) 2010-08-10 US disclosed
US-20090177010-A1 PROCESS OF MAKING SERTRALINE FORM I HETERO DRUGS LIMITED (IN) 2009-07-09 US disclosed
EP-0030081-A1 Antidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine and pharmaceutical compositions thereof PFIZER INC. (US) 1981-06-10 EP disclosed
EP-0028901-A1 Antidepressant derivatives of trans-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine and pharmaceutical compositions thereof PFIZER INC. (US) 1981-05-20 EP disclosed
EP-0028901-A1 Antidepressant derivatives of trans-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine and pharmaceutical compositions thereof PFIZER INC. (US) 1981-05-20 EP disclosed
EP-0028901-A1 Antidepressant derivatives of trans-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine and pharmaceutical compositions thereof PFIZER INC. (US) 1981-05-20 EP disclosed
US-4045488-A ANTIDEPRESSANTS OR PSYCHOMOTOR STIMULANTS PFIZER INC. (US) 1977-08-30 US disclosed
US-4045488-A ANTIDEPRESSANTS OR PSYCHOMOTOR STIMULANTS PFIZER INC. (US) 1977-08-30 US disclosed
US-4029731-A TREATING DEPRESSION PFIZER INC. (US) 1977-06-14 US disclosed
US-4029731-A TREATING DEPRESSION PFIZER INC. (US) 1977-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090177010-A1 PROCESS OF MAKING SERTRALINE FORM I HTR5A, HTR2A, HTR2C SLC6A2 22/4885SLC6A4 6/4885SLC6A3 104/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.