SCHEMBL29676258

SCHEMBL29676258

CC(=O)NC(C)(C)c1nc(C)cs1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.58
CNR2 P34972 3/20 0.44
MAPT P10636 2/20 0.39
RAB9A P51151 5/20 0.36
NPC1 O15118 4/20 0.36
PDE4A P27815 1/20 0.36
ADORA1 P30542 1/20 0.36
HTR2B P41595 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ALOX15 P16050 1/20 0.36
GAA P10253 1/20 0.36
POLB P06746 2/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
PKM P14618 1/20 0.35
FDPS P14324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25311505 0.81 SSTR4 (0.41) SSTR4CNR2MAPTRAB9ANPC1
SCHEMBL25307825 0.79 SSTR4 (0.39) SSTR4CNR2ALOX15
SCHEMBL19724475 0.76 SSTR4 (0.47) SSTR4CNR2MAPTRAB9ANPC1
SCHEMBL16366984 0.75 SSTR4 (0.43) SSTR4CNR2MAPTRAB9ANPC1
SCHEMBL16252613 0.74 SSTR4 (1.00) SSTR4
SCHEMBL19724971 0.74 SSTR4 (1.00) SSTR4
SCHEMBL634567 0.73 SSTR4 (0.43) SSTR4CNR2MAPTRAB9ANPC1
SCHEMBL132212 0.73 SSTR4 (0.44) SSTR4MAPTRAB9ANPC1PDE4A
SCHEMBL12817180 0.72 MAPK1 (0.56) SSTR4CNR2RAB9ANPC1POLB
SCHEMBL13151611 0.71 SSTR4 (0.43) SSTR4MAPTRAB9ANPC1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617166-B Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-05-17 CN claimed
CN-114948963-B Benzolactam compounds as protein kinase inhibitors 大冢制药株式会社 2025-05-27 CN disclosed
CN-114948963-A Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-08-30 CN disclosed
CN-108617166-B Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-05-17 CN disclosed