SCHEMBL29679782

SCHEMBL29679782

CC(C)(C)OC(=O)N1C[C@H](CO[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)OC[C@](C)(O)C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RORC P51449 10/20 0.41
SMYD2 Q9NRG4 2/20 0.37
SCD5 Q86SK9 1/20 0.36
GAA P10253 1/20 0.36
THRB P10828 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GPR119 Q8TDV5 1/20 0.35
EPHA2 P29317 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
NAMPT P43490 1/20 0.35
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29680582 1.00 RORC (0.41) RORCSMYD2SCD5GAATHRB
SCHEMBL29080094 0.90 SMYD2 (0.39) SMYD2SMN1; SMN2
SCHEMBL553857 0.84 EPHA2 (0.45) GAATHRBSMN1; SMN2GPR119EPHA2
SCHEMBL553856 0.84 EPHA2 (0.45) GAATHRBSMN1; SMN2GPR119EPHA2
SCHEMBL30987202 0.84 NR1H2 (0.34) RORCTHRBSMN1; SMN2EPHA2KDM4E
SCHEMBL30987065 0.84 NR1H2 (0.34) RORCTHRBSMN1; SMN2EPHA2KDM4E
SCHEMBL30987095 0.82 RORC (0.42) RORCGAATHRBSMN1; SMN2GPR119
SCHEMBL31299244 0.82 NAMPT (0.37) RORCSMYD2GAATHRBSMN1; SMN2
SCHEMBL29680617 0.82 NAMPT (0.37) RORCSMYD2GAATHRBSMN1; SMN2
SCHEMBL31299259 0.81 NAMPT (0.37) RORCSMYD2GAATHRBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624033-B2 KRAS inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2026-05-12 US disclosed
EP-4735439-A1 KRAS INHIBITORS Bristol-Myers Squibb Company (US) 2026-05-06 EP disclosed
EP-4735440-A1 KRAS INHIBITORS Bristol-Myers Squibb Company (US) 2026-05-06 EP disclosed
US-20250250271-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2025-08-07 US disclosed
US-20250154148-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2025-05-15 US disclosed
WO-2025006962-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-01-02 WO disclosed
WO-2025006967-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-01-02 WO disclosed
EP-4262807-A1 AZAQUINAZOLINE PAN-KRAS INHIBITORS Mirati Therapeutics, Inc. (US) 2023-10-25 EP disclosed
WO-2022132200-A1 AZAQUINAZOLINE PAN-KRAS INHIBITORS Mirati Therapeutics, Inc. (US) 2022-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250154148-A1 KRAS INHIBITORS KRAS, NRAS, HRAS RORC 2272/4885SMYD2 1603/4885SCD5 4238/4885
US-20250250271-A1 KRAS INHIBITORS KRAS, NRAS, HRAS RORC 2272/4885SMYD2 1603/4885SCD5 4238/4885
US-12624033-B2 KRAS inhibitors KRAS, NRAS, BRAF RORC 3778/4885SMYD2 2034/4885SCD5 4425/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.