SCHEMBL29680655

SCHEMBL29680655

O=Cc1ccc(-c2nc(Cl)nc3c2ccn3-c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.38
KDM4E B2RXH2 6/20 0.38
LMNA P02545 2/20 0.36
GLA P06280 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 1/20 0.35
ATM Q13315 1/20 0.34
OPRK1 P41145 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 2/20 0.33
CTDSP1 Q9GZU7 1/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PTGS2 P35354 1/20 0.33
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528679 1.00 ALDH1A1 (0.38) ALDH1A1KDM4ELMNAGLAHPGD
SCHEMBL29680579 0.95 ALDH1A1 (0.39) ALDH1A1KDM4ELMNAGLAHPGD
SCHEMBL24528625 0.95 ALDH1A1 (0.39) ALDH1A1KDM4ELMNAGLAHPGD
SCHEMBL16613450 0.87 KDM4E (0.45) ALDH1A1KDM4ELMNAGLAHPGD
SCHEMBL29516256 0.87 KDM4E (0.47) ALDH1A1KDM4ELMNAGLAHPGD
SCHEMBL16613618 0.87 KDM4E (0.47) ALDH1A1KDM4ELMNAGLAHPGD
SCHEMBL24528584 0.86 ALDH1A1 (0.37) ALDH1A1KDM4EMAPTATMKMT2A
SCHEMBL29681058 0.86 ALDH1A1 (0.37) ALDH1A1KDM4EMAPTATMKMT2A
SCHEMBL24528700 0.83 KDM4E (0.33) ALDH1A1KDM4ELMNAGLAHPGD
SCHEMBL29681072 0.83 KDM4E (0.33) ALDH1A1KDM4ELMNAGLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed