SCHEMBL29680966

SCHEMBL29680966

Clc1nc(Cl)c2ccn(-c3ccccc3)c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
POLB P06746 2/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
BIRC5 O15392 1/20 0.35
SRC P12931 1/20 0.35
NOTUM Q6P988 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
COMT P21964 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16613357 1.00 KDM4E (0.42) KDM4EPOLBCTDSP1HDAC1HDAC2
SCHEMBL4843924 0.86 BIRC5 (0.42) POLBHDAC1HDAC2BIRC5NOTUM
SCHEMBL21984170 0.85 NOTUM (0.40) KDM4EPOLBCTDSP1BIRC5SRC
SCHEMBL29516256 0.82 KDM4E (0.47) KDM4EPOLBCTDSP1CYP2D6CYP2C9
SCHEMBL16613618 0.82 KDM4E (0.47) KDM4EPOLBCTDSP1CYP2D6CYP2C9
SCHEMBL24528623 0.80 ALDH1A1 (0.41) KDM4EPOLBHDAC1HDAC2NPSR1
SCHEMBL29680986 0.80 ALDH1A1 (0.41) KDM4EPOLBHDAC1HDAC2NPSR1
SCHEMBL16613450 0.80 KDM4E (0.45) KDM4EPOLBCTDSP1CYP2D6CYP2C9
SCHEMBL16613668 0.76 KDM4E (0.41) KDM4EPOLBCTDSP1CYP2D6CYP2C9
SCHEMBL20351707 0.76 SRC (0.51) KDM4ETSHRCYP2C19SRCKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed