SCHEMBL29689641

SCHEMBL29689641

CNS(=O)(=O)c1ccc2c(c1)C(=Cc1[nH]c(C)c(CCCN3CCOCC3)c1C)C(=O)N2

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SRC P12931 16/20 0.74
KDR P35968 12/20 0.74
FGFR1 P11362 11/20 0.74
PDGFRB P09619 10/20 0.74
LCK P06239 9/20 0.74
FYN P06241 9/20 0.74
YES1 P07947 9/20 0.74
MET P08581 1/20 0.69
EGFR P00533 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5410964 0.87 KDR (0.60) SRCKDRFGFR1PDGFRBLCK
SCHEMBL6390071 0.86 SRC (0.68) SRCKDRFGFR1PDGFRBLCK
SCHEMBL6390067 0.86 SRC (0.68) SRCKDRFGFR1PDGFRBLCK
SCHEMBL4407079 0.85 KDR (0.66) SRCKDRFGFR1PDGFRBLCK
SCHEMBL4407081 0.85 KDR (0.66) SRCKDRFGFR1PDGFRBLCK
SCHEMBL6696492 0.85 SRC (0.98) SRCKDRFGFR1PDGFRBLCK
SCHEMBL5408957 0.83 MET (0.64) SRCKDRFGFR1PDGFRBLCK
SCHEMBL5408966 0.83 MET (0.64) SRCKDRFGFR1PDGFRBLCK
SCHEMBL4404881 0.83 KDR (0.82) SRCKDRFGFR1PDGFRBLCK
SCHEMBL4404878 0.83 KDR (0.82) SRCKDRFGFR1PDGFRBLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4562010-A1 CRYSTALLINE FORMS OF AN AKR1C3 DEPENDENT KARS INHIBITOR Novartis AG (CH) 2025-06-04 EP disclosed
WO-2024023666-A1 CRYSTALLINE FORMS OF AN AKR1C3 DEPENDENT KARS INHIBITOR NOVARTIS AG (CH) 2024-02-01 WO disclosed
EP-4007592-A1 ANGIOTENSIN TYPE 2 (AT2) RECEPTOR AGONISTS FOR USE IN THE TREATMENT OF CANCER LanthioPep B.V. (NL) 2022-06-08 EP disclosed