SCHEMBL29690171

SCHEMBL29690171

C=C(C)c1c(C)nc2ccc(Br)cn12

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHB3 P54753 1/20 0.51
GAA P10253 2/20 0.50
ALDH1A1 P00352 4/20 0.46
POLB P06746 3/20 0.46
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
NPC1 O15118 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
G6PD P11413 1/20 0.42
TSHR P16473 1/20 0.40
MAPK10 P53779 1/20 0.40
RXFP1 Q9HBX9 1/20 0.36
PSD A5PKW4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256814 0.84 KMT2A (0.58) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL8312175 0.81 EPHB3 (0.49) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL954716 0.81 EPHB3 (0.57) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL954299 0.79 EPHB3 (0.56) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL953778 0.79 EPHB3 (0.50) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL12850522 0.79 EPHB3 (0.60) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL29689941 0.78 ALDH1A1 (0.39) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL975608 0.75 GAA (0.58) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL18766608 0.75 EPHB3 (0.58) EPHB3GAAALDH1A1POLBKDM4E
SCHEMBL6223693 0.75 MAPK1 (0.63) EPHB3ALDH1A1POLBKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114605390-B Compounds having CDK kinase inhibitory activity, pharmaceutical compositions and uses thereof 上海凌达生物医药有限公司 2024-08-16 CN disclosed
CN-114605390-A Compound with CDK kinase inhibitory activity, pharmaceutical composition and use thereof 上海凌达生物医药有限公司 2022-06-10 CN disclosed